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Total posts by Rafał Kurczab: 4
publication
·
2 years ago
Low-basicity 5-HT7 Receptor Agonists Synthesized Using the van Leusen Multicomponent Protocol
by
Katarzyna Kiec-Kononowicz
,
Rafał Kurczab
,
Andrzej J. Bojarski
,
Jakub Staron
,
Grzegorz Satala
,
Ryszard Bugno
,
Adam S. Hogendorf
,
Agata Hogendorf
,
Tomasz Lenda
,
Maria Walczak
,
Gniewomir Latacz
,
Jadwiga Handzlik
,
Joanna M. Wieronska
,
Monika Wozniak
,
Paulina Cieslik
(
Jagiellonian University Medical College
,
Polish Academy of Sciences
)
publication
·
2 years ago
Halogen bonding enhances activity in a series of dual 5-HT6/D2 ligands designed in a hybrid bioisostere generation/virtual screening protocol
by
Rafał Kurczab
,
Andrzej J. Bojarski
,
Jakub Staron
,
Dawid Warszycki
,
Grzegorz Satala
,
Ryszard Bugno
,
Adam Hogendorf
(
Institute of Pharmacology Polish Academy of Sciences
,
Institute of Pharmacology PAS
)
publication
·
2 years ago
New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT7 and 5-HT1A receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies
by
Rafał Kurczab
,
Sebastiano Intagliata
,
Maria N. Modica
,
Valeria Pittalà
,
Loredana Salerno
,
Maria A. Siracusa
,
Alfredo Cagnotto
,
Mario Salmona
,
Giuseppe Romeo
(
Università di Catania
,
Polish Academy of Sciences
)
publication
·
2 years ago
Identification of Novel Serotonin Transporter Compounds by Virtual Screening
by
Mari Gabrielsen
,
Rafał Kurczab
,
Agata Siwek
,
Małgorzata Wolak
,
Aina W. Ravna
,
Kurt Kristiansen
,
Irina Kufareva
,
Ruben Abagyan
,
Gabriel Nowak
,
Zdzisław Chilmonczyk
,
Ingebrigt Sylte
,
Andrzej J. Bojarski
(
The Arctic University of Norway
)