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Total posts by University of Oxford: 5

publication · 2 months ago
In Silico Fragment-Based Design Identifies Subfamily B1 Metallo-B- lactamase Inhibitors
by Christopher J. Schofield, Colin W. G. Fishwick, Ricky Cain, Jurgen Brem, David Zollman, Michael A. McDonough, Rachel M. Johnson, James Spencer, Anne Makena, Martine I. Abboud, Samuel Cahill, Sook Y. Lee, Peter J. McHugh (University of Leeds, University of Oxford, University of Bristol, John Radcliffe Hospital)
publication · 3 years ago
Scaffold Hopping with Virtual Screening from IP3 to a Drug-Like Partial Agonist of the Inositol Trisphosphate Receptor
by Sridar R. Vasudevan, Nisha Singh, Grant C. Churchill (University of Oxford)
publication · 6 years ago
New potent dual inhibitors of CK2 and Pim kinases: Discovery and structural insight
by Renaud Prudent, Virginie Moucadel, Liliane Mouawad, Caroline Barette, Frederic Schmidt, Claude Cochet, Miriam López-Ramos, David Grierson, Jean-Claude Florent, Laurence Lafanechère, Jean-Baptiste Reiser, Céline F Sautel, Panagis Filippakopoulos, Alex N. Bullock, Stefan Knapp (University of Oxford, Université Paris-Sud, Centre National pour la Recherche Scientifique (CNRS), Unité Mixte de Recherche, Institut National de la Santé et de la Recherche Médicale (INSERM), Commissariat à l’énergie atomique (CEA), Partnership for Structural Biology, Université Joseph Fourier, Institut de Biologie Structurale Jean-Pierre Ebel (IBS), Institut Curie)
publication · 6 years ago
A specific two-pore domain potassium channel blocker defines the structure of the TASK-1 open pore
by Anne K. Streit, Michael F. Netter, Franca Kempf, Magdalena Walecki, Susanne Rinné, Murali K. Bollepalli, Regina Preisig-Müller, Vijay Renigunta, Jürgen Daut, Thomas Baukrowitz, Mark Sansom, Phillip J. Stansfeld, Niels Decher (University of Oxford, University of Marburg, University of Jena, University of Kiel)
publication · 7 years ago
Synthesis and Evaluation of 3-(Dihydroxyboryl)benzoic Acids as d,d-Carboxypeptidase R39 Inhibitors
by Steven R. Inglis, Astrid Zervosen, Esther C. Y. Woon, Thomas Gerards, Nathalie Teller, Delphine S. Fischer, André Luxen, Christopher J. Schofield (University of Oxford)