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Total posts by Brad E. Sleebs: 3

publication · 3 months ago
Enhanced antimalarial activity of plasmepsin V inhibitors by modification of the P2 position of PEXEL peptidomimetics
by Brad E. Sleebs, Matthew T. O’Neill, Alan F. Cowman, Justin A. Boddey, Kate E. Jarman, William Nguyen, Anthony N. Hodder, Richard Bestel de Lezongard, Peter E. Czabotar, Jennifer K. Thompson, Helene Jousset Sabroux (The University of Melbourne)
publication · 1 year ago
Optimization of 2-Anilino 4-Amino Substituted Quinazolines into Potent Antimalarial Agents with Oral in Vivo Activity
by Brad E. Sleebs, Alan F. Cowman, Paul R. Gilson, Cyrus Tan, Kate E. Jarman, Kym N. Lowes, Joan M. Curtis, William Nguyen, Adrian E. Di Rago, Hayley E. Bullen, Boris Prinz, Sandra Duffy, Jonathan B. Baell, Craig A. Hutton, Helene Jousset Subroux, Brendan S. Crabb, Vicky M. Avery (Griffith University, Monash University, University of Melbourne, The Walter and Eliza Hall Institute of Medical Research, Macfarlane Burnet Institute for Medical Research and Public Health)
publication · 1 year ago
Transition State Mimetics of the Plasmodium Export Element Are Potent Inhibitors of Plasmepsin V from P. falciparum and P. vivax
by Brad E. Sleebs, Michelle Gazdik, Matthew T. O’Neill, Pravin Rajasekaran, Sash Lopaticki, Kurt Lackovic, Kym Lowes, Brian J. Smith, Alan F. Cowman, Justin A. Boddey (The Walter and Eliza Hall Institute of Medical Research, The University of Melbourne)